Synthesis of Sterically Hindered α-Aminonitriles through 1,6-Aza-conjugate Addition of Anilines to δ-Cyano Substituted para-Quinone Methides
نویسندگان
چکیده
منابع مشابه
Practical catalytic method for synthesis of sterically hindered anilines.
A practical catalytic method for the synthesis of sterically hindered anilines is described. The amination of aryl and heteroaryl boronic esters is accomplished using a catalyst prepared in situ from commercially available and air-stable copper(i) triflate and diphosphine ligand. For the first time, the method can be applied to the synthesis of both secondary and tertiary anilines in the presen...
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ژورنال
عنوان ژورنال: Chinese Journal of Organic Chemistry
سال: 2020
ISSN: 0253-2786
DOI: 10.6023/cjoc202004027